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Indisetron Dihydrochloride

Tier C — Watch / trade

Indisetron Dihydrochloride

Kyorin Pharmaceutical Co Ltd
Originator
2004
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:5-HT3

Brand:Sinseron

Indications (approved):Nausea, 呕吐, Chemotherapy-induced nausea and vomiting

Regional status

US
-
EU
-
China
Phase II
2017-06-30
Japan
Withdrawn

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 4 · Total yield 0.4 g
INDI-0017252-83-7INDI-00256548-04-0INDI-003542-05-2INDI-004141549-84-0INDI-005—INDI-00672083-74-0API · Indisetron Dihydrochloride
CodeCAS No.Intermediate
INDI-0017252-83-7Available2-bromo-1,1-dimethoxyethane
INDI-00256548-04-0bis(2,2-dimethoxyethyl)amine
INDI-003542-05-23-oxopentanedioic acid
INDI-004141549-84-0(1R,5S)-3,9-dimethyl-3,9-diazabicyclo[3.3.1]nonan-7-one
INDI-005-(1R,5S,7s)-3,9-dimethyl-3,9-diazabicyclo[3.3.1]nonan-7-amine
INDI-00672083-74-01H-indazole-3-carbonyl chloride

Frequently asked questions

What are the approved indications of Indisetron Dihydrochloride?

Approved indications include: Nausea, 呕吐, Chemotherapy-induced nausea and vomiting.

When does the Indisetron Dihydrochloride patent expire?

No public expiry year is available for Indisetron Dihydrochloride yet; this page updates once verified.

How many synthesis routes are recorded for Indisetron Dihydrochloride?

1 synthesis routes are recorded; the shortest is 4 steps with 0.4 g total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Indisetron Dihydrochloride intermediates?

1 intermediate CAS of Indisetron Dihydrochloride are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Indisetron Dihydrochloride intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-09