Brilaroxazine
Tier C — Watch / tradeBrilaroxazine
Targets：5-HT1A, DRD4, DRD3, DRD2, 5-HT7, 5-HT6, 5-HT2A
Indications (approved)：Schizophrenia, Major depressive disorder, Pulmonary arterial hypertension, Idiopathic pulmonary fibrosis, Mania, Attention deficit hyperactivity disorder, Psoriasis
Regional status
Synthetic routes & intermediates1 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| RP-5063 | - | - |
| RP-5063-001 | 1568-70-3Available | 4-methoxy-2-nitrophenol |
| RP-5063-002 | 109364-95-6Available | ethyl 2-(4-methoxy-2-nitrophenoxy)acetate |
| RP-5063-003 | 103942-21-8Available | ethyl 2-(4-hydroxy-2-nitrophenoxy)acetate |
| RP-5063-004 | 110-52-1Available | 1,4-dibromobutane |
| RP-5063-005 | 1197155-12-6Available | ethyl 2-(4-(4-bromobutoxy)-2-nitrophenoxy)acetate |
| RP-5063-006 | 119532-26-2Available | 1-(2,3-dichlorophenyl)piperazine hydrochloride |
| RP-5063-007 | 1239729-01-1Available | ethyl 2-(4-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butoxy)-2-nitrophenoxy)acetate |
| RP-5063-008 | 1239729-06-6Available | 6-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butoxy)-2H-benzo[b][1,4]oxazin-3(4H)-one |
Frequently asked questions
What are the approved indications of Brilaroxazine?
Approved indications include: Schizophrenia, Major depressive disorder, Pulmonary arterial hypertension, Idiopathic pulmonary fibrosis, Mania, Attention deficit hyperactivity disorder, Psoriasis.
When does the Brilaroxazine patent expire?
No public expiry year is available for Brilaroxazine yet; this page updates once verified.
How many synthesis routes are recorded for Brilaroxazine?
1 synthesis routes are recorded; the shortest is 6 steps with 0.28 g total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Brilaroxazine intermediates?
8 intermediate CAS of Brilaroxazine are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.
How do I get a quote for Brilaroxazine intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-10-05