Taniborbactam
Tier C — Watch / tradeTaniborbactam
Targets：Beta Lactamase
Indications (approved)：Urinary tract infection, Pyelonephritis
Regional status
Synthetic routes & intermediates2 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| Tani-001 | 26507-91-5 | 2-methoxy-3-methylbenzoic acid |
| Tani-002 | 2377377-83-6 | tert-butyl 2-methoxy-3-methylbenzoate |
| Tani-003 | 2377377-87-0 | tert-butyl 3-(bromomethyl)-2-methoxybenzoate |
| Tani-004 | 1613269-60-5 | Benzoic acid, 3-[[(3aR,4R,6R,7aS)-hexahydro-3a,5,5-trimethyl-4,6-methano-1,3,2-benzodioxaborol-2-yl]methyl]-2-methoxy-, 1,1-dimethylethyl ester |
| Tani-005 | 2407879-39-2 | Benzoic acid, 3-[(2S )-2-chloro-2-[(3aR ,4R ,6R ,7aS )-hexahydro-3a,5,5-trimethyl-4,6-methano-1,3,2-benzodioxaborol-2-yl]ethyl]-2- methoxy-, 1,1-dimethylethyl ester |
| Tani-006 | 2407879-41-6 | Benzoic acid, 3-[(2R )-2-amino-2-[(3aR ,4R ,6R ,7aS )-hexahydro-3a,5,5-trimethyl-4,6-methano-1,3,2-benzodioxaborol-2-yl]ethyl]-2- methoxy-, 1,1-dimethylethyl ester |
| Tani-007 | 1613269-64-9 | 2-((1r,4r)-4-(tert-butoxycarbonyl(2-(tert-butoxycarbonylamino)ethyl)amino)cyclohexyl)acetic acid |
| Tani-008 | 2407879-42-7 | tert-butyl 3-((R)-2-(2-((1r,4R)-4-((tert-butoxycarbonyl)(2-((tert-butoxycarbonyl)amino)ethyl)amino)cyclohexyl)acetamido)-2-((3aR,4R,6R,7aS)-3a,5,5-trimethylhexahydro-4,6-methanobenzo[d][1,3,2]dioxaborol-2-yl)ethyl)-2-methoxybenzoate |
| Tani-009 | 76308-28-6 | ethyl 2-((1r,4r)-4-aminocyclohexyl)acetate |
| Tani-010 | 39684-80-5 | tert-butyl (2-bromoethyl)carbamate |
| Tani-011 | 1613269-84-3 | ethyl 2-((1r,4r)-4-(2-(tert-butoxycarbonylamino)ethylamino)cyclohexyl)acetate |
| Tani-012 | 1613269-62-7 | ethyl 2-((1r,4r)-4-(tert-butoxycarbonyl(2-(tert-butoxycarbonylamino)ethyl)amino)cyclohexyl)acetate |
| Code | CAS No. | Intermediate |
|---|---|---|
| Tani-001 | 26507-91-5 | 2-methoxy-3-methylbenzoic acid |
| Tani-002 | 2377377-83-6 | tert-butyl 2-methoxy-3-methylbenzoate |
| Tani-003 | 2377377-87-0 | tert-butyl 3-(bromomethyl)-2-methoxybenzoate |
| Tani-004 | 1613269-60-5 | Benzoic acid, 3-[[(3aR,4R,6R,7aS)-hexahydro-3a,5,5-trimethyl-4,6-methano-1,3,2-benzodioxaborol-2-yl]methyl]-2-methoxy-, 1,1-dimethylethyl ester |
| Tani-006 | 2407879-41-6 | Benzoic acid, 3-[(2R )-2-amino-2-[(3aR ,4R ,6R ,7aS )-hexahydro-3a,5,5-trimethyl-4,6-methano-1,3,2-benzodioxaborol-2-yl]ethyl]-2- methoxy-, 1,1-dimethylethyl ester |
| Tani-013 | 189153-10-4 | 2-((1r,4r)-4-(tert-butoxycarbonylamino)cyclohexyl)acetic acid |
| Tani-014 | 1613269-02-5 | Benzoic acid, 3-[(2R)-2-[[2-[trans-4-[[(1,1-dimethylethoxy)carbonyl]amino]cyclohexyl]acetyl]amino]-2-[(3aS,4S,6S,7aR)-hexahydro-3a,5,5-trimethyl-4,6-methano-1,3,2-benzodioxaborol-2-yl]ethyl]-2-methoxy-, 1,1-dimethylethyl ester |
| Tani-015 | 1613267-37-0 | (S)-3-(2-((1r,4S)-4-aminocyclohexyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid |
| Tani-016 | 89711-08-0 | tert-butyl (2-oxoethyl)carbamate |
| Tani-017 | 1613269-16-1 | (S)-3-(2-((1r,4S)-4-(2-(tert-butoxycarbonylamino)ethylamino)cyclohexyl)acetamido)-2-hydroxy-3,4-dihydro-2H-benzo[e][1,2]oxaborinine-8-carboxylic acid |
Frequently asked questions
What are the approved indications of Taniborbactam?
Approved indications include: Urinary tract infection, Pyelonephritis.
When does the Taniborbactam patent expire?
No public expiry year is available for Taniborbactam yet; this page updates once verified.
How many synthesis routes are recorded for Taniborbactam?
2 synthesis routes are recorded; the shortest is 8 steps with / total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Taniborbactam intermediates?
All intermediates in Taniborbactam routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.
How do I get a quote for Taniborbactam intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-10-07