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Brimonidine Tartrate

Tier C — Watch / trade

Brimonidine Tartrate

Allergan
Originator
1996
First approval
-
Expiry (public)
$0.15B ▲
Peak sales
Small molecule
Type

Targets:ADRA2

Brand:Brimocon, Alphagan

Indications (approved):Rosacea, Ocular hypertension, Open-angle glaucoma

Regional status

US
Approved
1996-09-06
EU
Approved
2014-02-20
China
Approved
1999-09-17
Japan
Approved
2012-01-18

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 4 · Total yield /
BRIM-0016298-37-9BRIM-00259803-96-2BRIM-003134892-46-9API · Brimonidine Tartrate
CodeCAS No.Intermediate
BRIM-0016298-37-9quinoxalin-6-amine
BRIM-00259803-96-25-bromoquinoxalin-6-amine hydrobromide
BRIM-003134892-46-95-bromo-6-isothiocyanatoquinoxaline

Frequently asked questions

What are the approved indications of Brimonidine Tartrate?

Approved indications include: Rosacea, Ocular hypertension, Open-angle glaucoma.

When does the Brimonidine Tartrate patent expire?

No public expiry year is available for Brimonidine Tartrate yet; this page updates once verified.

How many synthesis routes are recorded for Brimonidine Tartrate?

1 synthesis routes are recorded; the shortest is 4 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Brimonidine Tartrate intermediates?

All intermediates in Brimonidine Tartrate routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Brimonidine Tartrate intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-04