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Triptorelin Pamoate

Tier C — Watch / trade

Triptorelin Pamoate

Actavis A/S
Originator
2000
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:GnRHR

Brand:Trelstar (pamoate salt), Moapar (pamoate salt), Salvacyl, Trelstar LA, Trelstar Depot (pamoate salt), Trellasar (pamoate salt), Decapeptyl SR (pamoate salt), Pamorelin LA (pamoate salt)

Indications (approved):性早熟, Prostate cancer

Regional status

US
Approved
2000-06-15
EU
Discontinued
2007-10-01
China
Approved
2008-12-19
Japan
-

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 11 · Total yield 80 mg
TRIP-001—TRIP-002—TRIP-003—TRIP-004—TRIP-005—TRIP-006—TRIP-007—TRIP-008—TRIP-009—TRIP-010—TRIP-011—API · Triptorelin Pamoate
CodeCAS No.Intermediate
TRIP-001-methanamine
TRIP-002-2-amino-N-methylacetamide
TRIP-003-(S)-N-(2-(methylamino)-2-oxoethyl)pyrrolidine-2-carboxamide
TRIP-004-(S)-N-(2-(methylamino)-2-oxoethyl)-1-(Nw-tosyl-L-arginyl)pyrrolidine-2-carboxamide
TRIP-005-(S)-1-((S)-2-((S)-2-amino-4-methylpentanamido)-5-(3-tosylguanidino)pentanoyl)-N-(2-(methylamino)-2-oxoethyl)pyrrolidine-2-carboxamide
TRIP-006-(S)-1-(N2-L-tryptophyl-L-leucyl-Nw-tosyl-L-arginyl)-N-(2-(methylamino)-2-oxoethyl)pyrrolidine-2-carboxamide
TRIP-007--
TRIP-008--
TRIP-009--
TRIP-010--
TRIP-011--

Frequently asked questions

What are the approved indications of Triptorelin Pamoate?

Approved indications include: 性早熟, Prostate cancer.

When does the Triptorelin Pamoate patent expire?

No public expiry year is available for Triptorelin Pamoate yet; this page updates once verified.

How many synthesis routes are recorded for Triptorelin Pamoate?

1 synthesis routes are recorded; the shortest is 11 steps with 80 mg total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Triptorelin Pamoate intermediates?

All intermediates in Triptorelin Pamoate routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Triptorelin Pamoate intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-29