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Pimasertib hydrochloride

Tier C — Watch / trade

Pimasertib hydrochloride

Santhera Pharmaceuticals
Originator
-
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:MEK2, MEK1

Indications (approved):脑癌, Solid tumour, Non-small cell lung cancer, Lung cancer, Melanoma, Lymphoma, Brain metastases, 皮肤黑色素瘤

Regional status

US
Discontinued
2009-09-30
EU
Discontinued
2009-09-30
China
-
Japan
Discontinued
2012-09-30

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 2 · Total yield /
PIMAS-001393-53-3PIMAS-00229632-74-4PIMAS-003885588-03-4PIMAS-00461278-21-5API · Pimasertib hydrochloride
CodeCAS No.Intermediate
PIMAS-001393-53-33-fluoroisonicotinic acid
PIMAS-00229632-74-4Available2-fluoro-4-iodoaniline
PIMAS-003885588-03-43-((2-fluoro-4-iodophenyl)amino)isonicotinic acid
PIMAS-00461278-21-5(S)-3-aminopropane-1,2-diol

Frequently asked questions

What are the approved indications of Pimasertib hydrochloride?

Approved indications include: 脑癌, Solid tumour, Non-small cell lung cancer, Lung cancer, Melanoma, Lymphoma, Brain metastases, 皮肤黑色素瘤.

When does the Pimasertib hydrochloride patent expire?

No public expiry year is available for Pimasertib hydrochloride yet; this page updates once verified.

How many synthesis routes are recorded for Pimasertib hydrochloride?

1 synthesis routes are recorded; the shortest is 2 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Pimasertib hydrochloride intermediates?

1 intermediate CAS of Pimasertib hydrochloride are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Pimasertib hydrochloride intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-21