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Ensartinib Hydrochloride

Tier C — Watch / trade

Ensartinib Hydrochloride

Xcovery
Originator
2020
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets：ALK, c-Met, ROS

Brand：ENSACOVE

Indications (approved)：Non-small cell lung cancer

Regional status

US
Approved
2024-12-18
EU
Phase III
2016-06-01
China
Approved
2020-11-17
Japan
-

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 11 · Total yield 31 mg
ENSAR-001141-30-0ENSAR-0025469-69-2ENSAR-003446273-59-2ENSAR-004756520-66-8ENSAR-0051370651-29-8ENSAR-0061370651-32-3ENSAR-0071370651-34-5ENSAR-0081370651-36-7ENSAR-009619-45-4ENSAR-010—ENSAR-011—ENSAR-0122304609-25-2ENSAR-013—ENSAR-014756520-66-8API · Ensartinib Hydrochloride
CodeCAS No.Intermediate
ENSAR-001141-30-0Available3,6-dichloropyridazine
ENSAR-0025469-69-2Available6-chloropyridazin-3-amine
ENSAR-003446273-59-2Available4-bromo-6-chloropyridazin-3-amine
ENSAR-004756520-66-8Available1-(2,6-dichloro-3-fluorophenyl)ethan-1-ol
ENSAR-0051370651-29-8(R)-6-chloro-4-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)pyridazin-3-amine
ENSAR-0061370651-32-3-
ENSAR-0071370651-34-5-
ENSAR-0081370651-36-7-
ENSAR-009619-45-4methyl 4-aminobenzoate
ENSAR-010--
ENSAR-011--
ENSAR-0122304609-25-2(2R,6S)-2,6-dimethylpiperazine
ENSAR-013--
ENSAR-014756520-66-8Available1-(2,6-dichloro-3-fluorophenyl)ethan-1-ol

Frequently asked questions

What are the approved indications of Ensartinib Hydrochloride?

Approved indications include: Non-small cell lung cancer.

When does the Ensartinib Hydrochloride patent expire?

No public expiry year is available for Ensartinib Hydrochloride yet; this page updates once verified.

How many synthesis routes are recorded for Ensartinib Hydrochloride?

1 synthesis routes are recorded; the shortest is 11 steps with 31 mg total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Ensartinib Hydrochloride intermediates?

4 intermediate CAS of Ensartinib Hydrochloride are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Ensartinib Hydrochloride intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-29