Aminoarteether Maleate

Tier C — Watch / trade

Originator

First approval

Expiry (public)

No sales data

Peak sales

Small molecule

Type

Targets：Not applicable

Indications (approved)：Systemic lupus erythematosus

Regional status

China

Phase II

2019-07-24

Japan

Synthetic routes & intermediates1 routes

Originator routes × 0Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OptimisedRoute 1Steps 4 · Total yield 119 mg (Aminoarteether)

Aminoarteether-00163968-64-9Aminoarteether-002131175-87-6Aminoarteether-003101834-30-4Aminoarteether-0041289097-61-5Aminoarteether133162-24-0API · Aminoarteether Maleate

Code	CAS No.	Intermediate
Aminoarteether-001	63968-64-9	(3R,5aS,6R,8aS,9R)-3,6,9-trimethyloctahydro-3H-3,12-epoxy[1,2]dioxepino[4,3-i]isochromen-10(12H)-one
Aminoarteether-002	131175-87-6	(3R,5aS,6R,8aS,9R)-3,6,9-trimethyldecahydro-3H-3,12-epoxy[1,2]dioxepino[4,3-i]isochromen-10-ol
Aminoarteether-003	101834-30-4	(3R,5aS,6R,8aS,9R,10S)-10-(2-bromoethoxy)-3,6,9-trimethyldecahydro-3H-3,12-epoxy[1,2]dioxepino[4,3-i]isochromene
Aminoarteether-004	1289097-61-5	(3R,5aS,6R,8aS,9R,10S)-10-(2-azidoethoxy)-3,6,9-trimethyldecahydro-3H-3,12-epoxy[1,2]dioxepino[4,3-i]isochromene
Aminoarteether	133162-24-0	Ethanamine, 2-[[(3R,5aS,6R,8aS,9R,10S,12R,12aR)-decahydro-3,6,9-trimethyl-3,12-epoxy-12H-pyrano[4,3-j]-1,2-benzodioxepin-10-yl]oxy]-

Frequently asked questions

What are the approved indications of Aminoarteether Maleate?

Approved indications include: Systemic lupus erythematosus.

When does the Aminoarteether Maleate patent expire?

No public expiry year is available for Aminoarteether Maleate yet; this page updates once verified.

How many synthesis routes are recorded for Aminoarteether Maleate?

1 synthesis routes are recorded; the shortest is 4 steps with 119 mg (Aminoarteether) total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Aminoarteether Maleate intermediates?

All intermediates in Aminoarteether Maleate routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Aminoarteether Maleate intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-07