Carteolol Hydrochloride

Tier C — Watch / trade

AbbVie

Originator

1980

First approval

Expiry (public)

No sales data

Peak sales

Small molecule

Type

Targets：ADRB2, ADRB1

Brand：Mikelan LA, Mikelan, Arteolol, Carteol, Arteoptic, Teoptic, Cartrol, Ocupress

Indications (approved)：Hypertension, Ocular hypertension, Glaucoma, Angina pectoris, Arrhythmia

Regional status

China

Approved

1995-01-01

Japan

Approved

1980-10-25

Synthetic routes & intermediates3 routes

Originator routes × 0Optimised (non-patent) × 3Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OptimisedRoute 1Steps 4 · Total yield /

Carteolol Hydrochloride-001108-46-3Carteolol Hydrochloride-002504-02-9Carteolol Hydrochloride-0035220-49-5Carteolol Hydrochloride-00479-10-7Carteolol Hydrochloride-0055057-12-5Carteolol Hydrochloride-00630389-33-4API · Carteolol Hydrochloride

Code	CAS No.	Intermediate
Carteolol Hydrochloride-001	108-46-3	Benzene-1,3-diol
Carteolol Hydrochloride-002	504-02-9	1,3-Cyclohexanedione
Carteolol Hydrochloride-003	5220-49-5	3-Aminocyclohex-2-en-1-one
Carteolol Hydrochloride-004	79-10-7	2-Propenoic acid
Carteolol Hydrochloride-005	5057-12-5	1,2,3,4,5,6,7,8-Octahydroquinoline-2,5-dione
Carteolol Hydrochloride-006	30389-33-4	5-Hydroxy-1,2,3,4-tetrahydroquinolin-2-one

OptimisedRoute 2Steps 5 · Total yield /

Carteolol Hydrochloride-00751781-14-7Carteolol Hydrochloride-01051781-13-6Carteolol Hydrochloride-008252267-77-9Carteolol Hydrochloride-00630389-33-4Carteolol Hydrochloride-01296-24-2Carteolol Hydrochloride-011106-89-8Carteolol Hydrochloride-0133132-64-7Carteolol Hydrochloride-00975-64-9API · Carteolol Hydrochloride

Code	CAS No.	Intermediate
Carteolol Hydrochloride-007	51781-14-7	5-(oxiran-2-ylmethoxy)-1,2,3,4-tetrahydroquinolin-2-one
Carteolol Hydrochloride-010	51781-13-6	5-(3-chloro-2-hydroxypropoxy)-1,2,3,4-tetrahydroquinolin-2-one
Carteolol Hydrochloride-008	252267-77-9	decahydroquinoline-2,5-dione
Carteolol Hydrochloride-006	30389-33-4	5-Hydroxy-1,2,3,4-tetrahydroquinolin-2-one
Carteolol Hydrochloride-012	96-24-2	(+/-)-2,3-Dihydroxychloropropane
Carteolol Hydrochloride-011	106-89-8	(+/-)-2-(Chloromethyl)oxirane
Carteolol Hydrochloride-013	3132-64-7	1-Bromo-2,3-epoxypropane
Carteolol Hydrochloride-009	75-64-9 Available	1,1-Dimethylethylamine

OptimisedRoute 3Steps 5 · Total yield /

Carteolol Hydrochloride-0141138-80-3Carteolol Hydrochloride-015506-59-2Carteolol Hydrochloride-016167303-60-8Carteolol Hydrochloride-0171857-19-8Carteolol Hydrochloride-01879-09-4Carteolol Hydrochloride-0191158271-30-7Carteolol Hydrochloride-020529-28-2Carteolol Hydrochloride-0211927901-90-3Carteolol Hydrochloride-0221927901-84-5API · Carteolol Hydrochloride

Code	CAS No.	Intermediate
Carteolol Hydrochloride-014	1138-80-3 Available	2-(Benzyloxycarbonylamino)acetic acid
Carteolol Hydrochloride-015	506-59-2 Available	Dimethylamine hydrochloride
Carteolol Hydrochloride-016	167303-60-8	Benzyl [2-(dimethylamino)-2-oxoethyl]carbamate
Carteolol Hydrochloride-017	1857-19-8	N,N-Dimethylglycinamide
Carteolol Hydrochloride-018	79-09-4 Available	Carboxyethane
Carteolol Hydrochloride-019	1158271-30-7	N-[2-(Dimethylamino)-2-oxoethyl]propanamide
Carteolol Hydrochloride-020	529-28-2	1-Iodo-2-methoxybenzene
Carteolol Hydrochloride-021	1927901-90-3	N-[2-(Dimethylamino)-2-oxoethyl]-3-(2-methoxyphenyl)propanamide
Carteolol Hydrochloride-022	1927901-84-5	2-(5-Methoxy-2-oxo-3,4-dihydroquinolin-1(2H)-yl)-N,N-dimethylacetamide

Frequently asked questions

What are the approved indications of Carteolol Hydrochloride?

Approved indications include: Hypertension, Ocular hypertension, Glaucoma, Angina pectoris, Arrhythmia.

When does the Carteolol Hydrochloride patent expire?

No public expiry year is available for Carteolol Hydrochloride yet; this page updates once verified.

How many synthesis routes are recorded for Carteolol Hydrochloride?

3 synthesis routes are recorded; the shortest is 4 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Carteolol Hydrochloride intermediates?

4 intermediate CAS of Carteolol Hydrochloride are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Carteolol Hydrochloride intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-29