Gildeuretinol

Tier C — Watch / trade

Gildeuretinol

Alkeus

Originator

First approval

Expiry (public)

No sales data

Peak sales

Small molecule

Type

Targets：Not applicable

Indications (approved)：Stargardt病, 地图状萎缩, 年龄相关性黄斑变性

Regional status

Phase III

2019-05-07

China

Japan

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 7 · Total yield 0.60g (ALK-001)

ALK-001-00179-77-6ALK-001-002867-13-0ALK-001-00317974-55-9ALK-001-0043917-39-3ALK-001-0053917-41-7ALK-001-0067379-29-5ALK-001-00786530-28-1ALK-001-00886561-74-2ALK-001-009118139-35-8API · Gildeuretinol

Code	CAS No.	Intermediate
ALK-001-001	79-77-6	(E)-4-(2,6,6-trimethylcyclohex-1-enyl)but-3-en-2-one
ALK-001-002	867-13-0 Available	ethyl 2-(diethoxyphosphoryl)acetate
ALK-001-003	17974-55-9	(2E,4E)-ethyl 3-methyl-5-(2,6,6-trimethylcyclohex-1-enyl)penta-2,4-dienoate
ALK-001-004	3917-39-3	(2Z,4E)-3-methyl-5-(2,6,6-trimethylcyclohex-1-en-1-yl)penta-2,4-dien-1-ol
ALK-001-005	3917-41-7	(2E,4E)-3-methyl-5-(2,6,6-trimethylcyclohex-1-en-1-yl)penta-2,4-dienal
ALK-001-006	7379-29-5	1,1,1-3D-Acetone
ALK-001-007	86530-28-1	(3E,5E,7E)- 20,20.20-trideutero-6-methyl-8-(2,6,6-trimethylcyclohex-1-enyl)octa-3,5,7-trien-2-one
ALK-001-008	86561-74-2	(2E,4E,6E,8E)-ethyl 20,20.20-trideutero-3,7-dimethyl-9-(2,6,6-trimethylcyclohex-1-enyl)nona-2,4,6,8-tetraenoate
ALK-001-009	118139-35-8	(2E,4E,6E,8E)-20,20.20-trideutero-3,7-dimethyl-9-(2,6,6-trimethylcyclohex-1-enyl)nona-2,4,6,8-tetraen-1-ol

Frequently asked questions

What are the approved indications of Gildeuretinol?

Approved indications include: Stargardt病, 地图状萎缩, 年龄相关性黄斑变性.

When does the Gildeuretinol patent expire?

No public expiry year is available for Gildeuretinol yet; this page updates once verified.

How many synthesis routes are recorded for Gildeuretinol?

1 synthesis routes are recorded; the shortest is 7 steps with 0.60g (ALK-001) total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Gildeuretinol intermediates?

1 intermediate CAS of Gildeuretinol are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Gildeuretinol intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-08