← Back to patent-cliff list

Yogliptin

Tier C — Watch / trade

Yogliptin

-
Originator
-
First approval
-
Expiry (public)
No sales data
Peak sales
-
Type

Targets:DPP4

Indications (approved):Type 2 diabetes

Regional status

US
-
EU
-
China
Phase III
2022-01-01
Japan
-

Synthetic routes & intermediates1 routes

Originator routes × 0Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OptimisedRoute 1Steps 4 · Total yield 153 mg (Yogliptin)
Yogliptin-00193703-24-3Yogliptin-0023355-28-0Yogliptin-003666816-98-4Yogliptin-004143163-70-6Yogliptin-0051518906-22-3Yogliptin-006309956-78-3Yogliptin-0071518906-26-7API · Yogliptin
CodeCAS No.Intermediate
Yogliptin-00193703-24-3Available8-bromo-3-methyl-3,7-dihydro-1H-purine-2,6-dione
Yogliptin-0023355-28-0Available1-bromobut-2-yne
Yogliptin-003666816-98-4Available8-bromo-7-(but-2-yn-1-yl)-3-methyl-3,7-dihydro-1H-purine-2,6-dione
Yogliptin-004143163-70-62-(bromomethyl)-5-fluorobenzo[d]thiazole
Yogliptin-0051518906-22-38-bromo-7-(but-2-yn-1-yl)-1-((5-fluorobenzo[d]thiazol-2-yl)methyl)-3-methyl-3,7-dihydro-1H-purine-2,6-dione
Yogliptin-006309956-78-3Availabletert-butyl (R)-piperidin-3-ylcarbamate
Yogliptin-0071518906-26-7tert-butyl (R)-(1-(7-(but-2-yn-1-yl)-1-((5-fluorobenzo[d]thiazol-2-yl)methyl)-3-methyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)piperidin-3-yl)carbamate

Frequently asked questions

What are the approved indications of Yogliptin?

Approved indications include: Type 2 diabetes.

When does the Yogliptin patent expire?

No public expiry year is available for Yogliptin yet; this page updates once verified.

How many synthesis routes are recorded for Yogliptin?

1 synthesis routes are recorded; the shortest is 4 steps with 153 mg (Yogliptin) total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Yogliptin intermediates?

4 intermediate CAS of Yogliptin are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Yogliptin intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-21