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Arterolane maleate/Piperaquine Phosphate

Tier C — Watch / trade

Arterolane maleate/Piperaquine Phosphate

Ranbaxy Laboratories Ltd., Beijing Representative Office
Originator
2012
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:CYP3A4

Brand:Synriam

Indications (approved):Plasmodium infection

Regional status

US
-
EU
-
China
-
Japan
-

Synthetic routes & intermediates1 routes

Originator routes × 0Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OptimisedRoute 1Steps 3 · Total yield 26.9(Piperaquine Phosphate (API))
Piperaquine Phosphate-001—Piperaquine Phosphate-002—Piperaquine Phosphate-003—Piperaquine Phosphate-0041143349-11-4Piperaquine Phosphate-005—Piperaquine Phosphate-0064085-31-8API · Arterolane maleate/Piperaquine Phosphate
CodeCAS No.Intermediate
Piperaquine Phosphate-001-4,7-Bis(chloranyl)quinoline
Piperaquine Phosphate-002-1,4-Diazacyclohexane
Piperaquine Phosphate-003-7-Chloro-4-(1-piperazinyl)quinoline
Piperaquine Phosphate-0041143349-11-47-Chloro-4-(piperazin-1-yl)quinoline hydrogen chloride
Piperaquine Phosphate-005-1,3-Dibromopropane
Piperaquine Phosphate-0064085-31-84,4'-(Propane-1,3-diyl)bis(piperazin-4,1-diy)bis(7-chloroquinoline)

Frequently asked questions

What are the approved indications of Arterolane maleate/Piperaquine Phosphate?

Approved indications include: Plasmodium infection.

When does the Arterolane maleate/Piperaquine Phosphate patent expire?

No public expiry year is available for Arterolane maleate/Piperaquine Phosphate yet; this page updates once verified.

How many synthesis routes are recorded for Arterolane maleate/Piperaquine Phosphate?

1 synthesis routes are recorded; the shortest is 3 steps with 26.9(Piperaquine Phosphate (API)) total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Arterolane maleate/Piperaquine Phosphate intermediates?

All intermediates in Arterolane maleate/Piperaquine Phosphate routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Arterolane maleate/Piperaquine Phosphate intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-29