Cenerimod
Tier C — Watch / tradeCenerimod
Targets：S1PR1
Indications (approved)：狼疮肾炎, Systemic lupus erythematosus, Renal impairment, Hepatic function decline
Regional status
Synthetic routes & intermediates1 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| - | - | - |
| - | 1694-31-1Available | tert-butyl 3-oxobutanoate |
| - | 110-52-1Available | 1,4-dibromobutane |
| - | 6004-60-0 | 1-cyclopentylethanone |
| - | 1368348-22-4 | 6-cyclopentyl-2-oxo-1,2-dihydropyridine-4-carboxylic acid |
| - | 1495273-79-4 | methyl 6-cyclopentyl-2-oxo-1,2-dihydropyridine-4-carboxylate |
| - | 1495273-80-7 | methyl 2-chloro-6-cyclopentylisonicotinate |
| - | 1122089-67-1 | 2-cyclopentyl-6-methoxyisonicotinic acid |
| - | 1150644-85-1 | (R)-4-((2,2-dimethyl-1,3-dioxolan-4-yl)methoxy)-3-ethyl-N-hydroxy-5-methylbenzimidamide |
| - | 1980852-81-0 | (R)-N-((2-cyclopentyl-6-methoxyisonicotinoyl)oxy)-4-((2,2-dimethyl-1,3-dioxolan-4-yl)methoxy)-3-ethyl-5-methylbenzimidamide |
| - | 1980852-82-1 | (R)-5-(2-cyclopentyl-6-methoxypyridin-4-yl)-3-(4-((2,2-dimethyl-1,3-dioxolan-4-yl)methoxy)-3-ethyl-5-methylphenyl)-1,2,4-oxadiazole |
| - | 4909-95-9 | 3-ethyl-4-hydroxy-5-methylbenzonitrile |
| - | 14347-78-5 | (R)-(2,2-dimethyl-1,3-dioxolan-4-yl)methanol |
Frequently asked questions
What are the approved indications of Cenerimod?
Approved indications include: 狼疮肾炎, Systemic lupus erythematosus, Renal impairment, Hepatic function decline.
When does the Cenerimod patent expire?
No public expiry year is available for Cenerimod yet; this page updates once verified.
How many synthesis routes are recorded for Cenerimod?
1 synthesis routes are recorded; the shortest is 9 steps with 3.3 kg total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Cenerimod intermediates?
2 intermediate CAS of Cenerimod are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.
How do I get a quote for Cenerimod intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-10-21