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Retagliptin Phosphate

Tier C — Watch / trade

Retagliptin Phosphate

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Originator
2023
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:DPP4

Indications (approved):Type 2 diabetes

Regional status

US
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EU
-
China
Approved
2023-06-27
Japan
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Factories producing this API3

Factories registered as producing this API in our sourcing network (RFQ records + product master), sorted by RFQ activity; the snapshot carries no cost or customer data.

3 producing factories on file — sign in to view the named list (factory details are not shown to guests).

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Synthetic routes & intermediates1 routes

Originator routes × 0Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OptimisedRoute 1Steps 9 · Total yield 5.90 g
RETAG-001209995-38-0RETAG-002108-59-8RETAG-003769195-26-8RETAG-00420989-17-7RETAG-0051338939-58-4RETAG-0061338939-59-5RETAG-0071338939-60-8RETAG-0081358715-37-3RETAG-0091598419-96-5RETAG-0101598419-97-6RETAG-011407-25-0RETAG-0121598419-90-9RETAG-0131598419-91-0API · Retagliptin Phosphate
CodeCAS No.Intermediate
RETAG-001209995-38-02-(2,4,5-trifluorophenyl)acetic acid
RETAG-002108-59-8Availabledimethyl malonate
RETAG-003769195-26-8methyl 3-oxo-4-(2,4,5-trifluorophenyl)butanoate
RETAG-00420989-17-7(S)-2-amino-2-phenylethanol
RETAG-0051338939-58-4(S,E)-methyl 3-((2-hydroxy-1-phenylethyl)amino)-4-(2,4,5-trifluorophenyl)but-2-enoate
RETAG-0061338939-59-5(S)-3-phenyl-5-(2,4,5-trifluorobenzyl)-3,4-dihydro-1,4-oxazepin-7(2H)-one
RETAG-0071338939-60-8(3S,5R)-3-phenyl-5-(2,4,5-trifluorobenzyl)-1,4-oxazepan-7-one
RETAG-0081358715-37-3methyl 3-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylate
RETAG-0091598419-96-5methyl 7-((R)-3-(((S)-2-hydroxy-1-phenylethyl)amino)-4-(2,4,5-trifluorophenyl)butanoyl)-3-(trifluoromethyl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxylate
RETAG-0101598419-97-6methyl 2-amino-2-(pyrazin-2-yl)acetate hydrochloride
RETAG-011407-25-02,2,2-trifluoroacetic anhydride
RETAG-0121598419-90-9methyl 2-(pyrazin-2-yl)-2-(2,2,2-trifluoroacetamido)acetate
RETAG-0131598419-91-0methyl 3-(trifluoromethyl)imidazo[1,5-a]pyrazine-1-carboxylate

Frequently asked questions

What are the approved indications of Retagliptin Phosphate?

Approved indications include: Type 2 diabetes.

When does the Retagliptin Phosphate patent expire?

No public expiry year is available for Retagliptin Phosphate yet; this page updates once verified.

How many synthesis routes are recorded for Retagliptin Phosphate?

1 synthesis routes are recorded; the shortest is 9 steps with 5.90 g total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Retagliptin Phosphate intermediates?

1 intermediate CAS of Retagliptin Phosphate are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Retagliptin Phosphate intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-29