Ganfeborole
Tier C — Watch / tradeGanfeborole
Targets：LARS
Indications (approved)：Pulmonary tuberculosis, Mycobacterium tuberculosis infection
Regional status
Synthetic routes & intermediates1 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| GSK-3036656-001 | 196081-71-7 | 2-bromo-3-hydroxybenzaldehyde |
| GSK-3036656-002 | 540-51-2 | 2-bromoethan-1-ol |
| GSK-3036656-003 | 1093644-11-1 | 2-bromo-3-(2-((tetrahydro-2H-pyran-2-yl)oxy)ethoxy)benzaldehyde |
| GSK-3036656-004 | 1093643-64-1 | 3-(2-((tetrahydro-2H-pyran-2-yl)oxy)ethoxy)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde |
| GSK-3036656-005 | 2131798-37-1 | 7-(2-hydroxyethoxy)-3-(nitromethyl)benzo[c][1,2]oxaborol-1(3H)-ol |
| GSK-3036656-006 | 2131798-39-3 | 4-chloro-7-(2-hydroxyethoxy)-3-(nitromethyl)benzo[c][1,2]oxaborol-1(3H)-ol |
| GSK-3036656-007 | 2131797-85-6 | 3-(aminomethyl)-4-chloro-7-(2-hydroxyethoxy)benzo[c][1,2]oxaborol-1(3H)-ol hydrochloride |
| GSK-3036656-008 | 2135692-04-3 | tert-butyl ((4-chloro-1-hydroxy-7-(2-hydroxyethoxy)-1,3-dihydrobenzo[c][1,2]oxaborol-3-yl)methyl)carbamate |
Frequently asked questions
What are the approved indications of Ganfeborole?
Approved indications include: Pulmonary tuberculosis, Mycobacterium tuberculosis infection.
When does the Ganfeborole patent expire?
No public expiry year is available for Ganfeborole yet; this page updates once verified.
How many synthesis routes are recorded for Ganfeborole?
1 synthesis routes are recorded; the shortest is 7 steps with 1.2 g total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Ganfeborole intermediates?
All intermediates in Ganfeborole routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.
How do I get a quote for Ganfeborole intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-10-08