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Gacyclidine

Tier C — Watch / trade

Gacyclidine

Ipsen Inc
Originator
-
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:NMDAR

Indications (approved):耳鸣

Regional status

US
Phase II
2019-04-04
EU
Phase II
2021-03-22
China
-
Japan
-

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 5 · Total yield 118 mg (Gacyclidine Hydrochloride)
GACYC-0015713-61-1GACYC-002583-60-8GACYC-003—GACYC-004—GACYC-005—GACYC-006111-24-0GACYC-007—Gacyclidine Hydrochloride68134-81-6API · Gacyclidine
CodeCAS No.Intermediate
GACYC-0015713-61-1thiophen-2-ylmagnesium bromide
GACYC-002583-60-82-methylcyclohexan-1-one
GACYC-003-(2S)-2-methyl-1-(thiophen-2-yl)cyclohexan-1-ol
GACYC-004-2-((2S)-1-azido-2-methylcyclohexyl)thiophene
GACYC-005-(2S)-2-methyl-1-(thiophen-2-yl)cyclohexan-1-amine
GACYC-006111-24-01,5-dibromopentane
GACYC-007-1-((2S)-2-methyl-1-(thiophen-2-yl)cyclohexyl)piperidine
Gacyclidine Hydrochloride68134-81-61-((1R,2S)-2-methyl-1-(thiophen-2-yl)cyclohexyl)piperidine hydrochloride

Frequently asked questions

What are the approved indications of Gacyclidine?

Approved indications include: 耳鸣.

When does the Gacyclidine patent expire?

No public expiry year is available for Gacyclidine yet; this page updates once verified.

How many synthesis routes are recorded for Gacyclidine?

1 synthesis routes are recorded; the shortest is 5 steps with 118 mg (Gacyclidine Hydrochloride) total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Gacyclidine intermediates?

All intermediates in Gacyclidine routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Gacyclidine intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-08