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Selatogrel

Tier C — Watch / trade

Selatogrel

Idorsia Pharmaceuticals Ltd
Originator
-
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:P2RY12

Indications (approved):Myocardial infarction, 慢性冠脉综合征, Hepatic function decline, Coronary artery lesion

Regional status

US
Phase III
2021-08-14
EU
Phase III
2021-08-14
China
Phase III
2021-08-14
Japan
Phase III
2021-08-14

Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 15 · Total yield /
ACT-246475—ACT-246475-00193267-04-0ACT-246475-002851475-17-7ACT-246475-0031159501-66-2ACT-246475-00450606-32-1ACT-246475-0051159501-70-8ACT-246475-0061159501-71-9ACT-246475-0071159501-69-5ACT-246475-0081159501-72-0ACT-246475-009592-34-7ACT-246475-0102759-28-6ACT-246475-0111019928-96-1ACT-246475-012100243-39-8ACT-246475-013101469-92-5ACT-246475-014550371-69-2ACT-246475-015685828-16-4ACT-246475-016913952-59-7ACT-246475-0171875708-16-9ACT-246475-018325685-59-4ACT-246475-019325685-75-4API · Selatogrel
CodeCAS No.Intermediate
ACT-246475--
ACT-246475-00193267-04-0Available(R)-methyl 2-((tert-butoxycarbonyl)amino)-3-iodopropanoate
ACT-246475-002851475-17-7(R)-methyl 2-((tert-butoxycarbonyl)amino)-3-(diethoxyphosphoryl)propanoate
ACT-246475-0031159501-66-2(R)-2-((tert-butoxycarbonyl)amino)-3-(diethoxyphosphoryl)propanoic acid
ACT-246475-00450606-32-1butyl piperazine-1-carboxylate
ACT-246475-0051159501-70-8(R)-butyl 4-(2-((tert-butoxycarbonyl)amino)-3-(diethoxyphosphoryl)propanoyl)piperazine-1-carboxylate
ACT-246475-0061159501-71-9(R)-butyl 4-(2-amino-3-(diethoxyphosphoryl)propanoyl)piperazine-1-carboxylate hydrochloride
ACT-246475-0071159501-69-5(S)-6-(3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carboxylic acid
ACT-246475-0081159501-72-0butyl 4-((R)-3-(diethoxyphosphoryl)-2-(6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carboxamido)propanoyl)piperazine-1-carboxylate
ACT-246475-009592-34-7butyl carbonochloridate
ACT-246475-0102759-28-61-benzylpiperazine
ACT-246475-0111019928-96-1butyl 4-benzylpiperazine-1-carboxylate
ACT-246475-012100243-39-8(S)-pyrrolidin-3-ol
ACT-246475-013101469-92-5(S)-tert-butyl 3-hydroxypyrrolidine-1-carboxylate
ACT-246475-014550371-69-2(S)-tert-butyl 3-methoxypyrrolidine-1-carboxylate
ACT-246475-015685828-16-4(S)-3-methoxypyrrolidine hydrochloride
ACT-246475-016913952-59-76-chloro-2-phenylpyrimidine-4-carboxylic acid
ACT-246475-0171875708-16-96-(methoxymethyl)-2-phenylpyrimidin-4-ol
ACT-246475-018325685-59-44-chloro-6-(methoxymethyl)-2-phenylpyrimidine
ACT-246475-019325685-75-4(6-chloro-2-phenylpyrimidin-4-yl)methanol

Frequently asked questions

What are the approved indications of Selatogrel?

Approved indications include: Myocardial infarction, 慢性冠脉综合征, Hepatic function decline, Coronary artery lesion.

When does the Selatogrel patent expire?

No public expiry year is available for Selatogrel yet; this page updates once verified.

How many synthesis routes are recorded for Selatogrel?

1 synthesis routes are recorded; the shortest is 15 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Selatogrel intermediates?

1 intermediate CAS of Selatogrel are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Selatogrel intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-06