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Filgotinib Maleate

Tier C — Watch / trade

Filgotinib Maleate

Galapagos Nv
Originator
2020
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:JAK1

Brand:Jyseleca

Indications (approved):Ulcerative colitis, Rheumatoid arthritis

Regional status

US
Phase III
2016-07-27
EU
Approved
2020-09-24
China
-
Japan
Approved
2020-09-25

Factories producing this API1

Factories registered as producing this API in our sourcing network (RFQ records + product master), sorted by RFQ activity; the snapshot carries no cost or customer data.

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Synthetic routes & intermediates2 routes

Originator routes × 1Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 6 · Total yield /
FILG-00119798-81-3FILG-00216182-04-0FILG-0031010120-59-8FILG-0041010120-55-4FILG-0054023-34-1FILG-0061142943-96-1FILG-00759016-93-2FILG-0081142936-49-9FILG-0091206163-59-8FILG-01039093-93-1API · Filgotinib Maleate
CodeCAS No.Intermediate
FILG-00119798-81-3Available6-bromopyridin-2-amine
FILG-00216182-04-0AvailableO-ethyl carbonisothiocyanatidate
FILG-0031010120-59-8Available-
FILG-0041010120-55-4Available-
FILG-0054023-34-1Availablecyclopropanecarbonyl chloride
FILG-0061142943-96-1AvailableN-(5-bromo-[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide
FILG-00759016-93-2Available(4-(hydroxymethyl)phenyl)boronic acid
FILG-0081142936-49-9Available-
FILG-0091206163-59-8Available-
FILG-01039093-93-1Availablethiomorpholine 1,1-dioxide
OptimisedRoute 2Steps 8 · Total yield /
FILG-00216182-04-0FILG-0054023-34-1FILG-01145644-21-1FILG-012159603-71-1FILG-013—FILG-0141819973-35-7FILG-0151092563-25-1FILG-0161819973-38-0FILG-0171819973-36-8FILG-0181819973-37-9FILG-0191257705-09-1API · Filgotinib Maleate
CodeCAS No.Intermediate
FILG-00216182-04-0AvailableO-ethyl carbonisothiocyanatidate
FILG-0054023-34-1Availablecyclopropanecarbonyl chloride
FILG-01145644-21-1Available-
FILG-012159603-71-1Available-
FILG-013-tert-butyl (6-hydroxypyridin-2-yl)carbamate
FILG-0141819973-35-7Available-
FILG-0151092563-25-1Available-
FILG-0161819973-38-0Available-
FILG-0171819973-36-8Available-
FILG-0181819973-37-9Available-
FILG-0191257705-09-1Available-

Frequently asked questions

What are the approved indications of Filgotinib Maleate?

Approved indications include: Ulcerative colitis, Rheumatoid arthritis.

When does the Filgotinib Maleate patent expire?

No public expiry year is available for Filgotinib Maleate yet; this page updates once verified.

How many synthesis routes are recorded for Filgotinib Maleate?

2 synthesis routes are recorded; the shortest is 6 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Filgotinib Maleate intermediates?

18 intermediate CAS of Filgotinib Maleate are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Filgotinib Maleate intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-29