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Talaporfin Sodium

Tier C — Watch / trade

Talaporfin Sodium

-
Originator
2003
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:Not applicable

Brand:Aptocine, Laserphyrin

Indications (approved):Lung cancer, 脑癌

Regional status

US
Discontinued
2003-10-01
EU
No progress
2006-07-01
China
Phase I
2009-02-04
Japan
Approved
2003-10-16

Synthetic routes & intermediates2 routes

Originator routes × 1Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 3 · Total yield /
TALAS-00119660-77-6TALAS-0021791-13-5TALAS-003—API · Talaporfin Sodium
CodeCAS No.Intermediate
TALAS-00119660-77-6-
TALAS-0021791-13-5(S)-di-tert-butyl 2-aminosuccinate hydrochloride
TALAS-003--
OptimisedRoute 2Steps 2 · Total yield /
TALAS-00119660-77-6TALAS-0041000783-47-0TALAS-00556-84-8API · Talaporfin Sodium
CodeCAS No.Intermediate
TALAS-00119660-77-6-
TALAS-0041000783-47-021H-9,12-Imino-2,22-metheno-7,4:14,17-dinitrilo-1H-oxepino[4,5-b]azacyclononadecine-16-propanoic acid, 10-ethenyl-5-ethyl-15,16,18,19-tetrahydro-6,11,15,23-tetramethyl-19,21-dioxo-, (15S,16S)-
TALAS-00556-84-8(S)-2-aminosuccinic acid

Frequently asked questions

What are the approved indications of Talaporfin Sodium?

Approved indications include: Lung cancer, 脑癌.

When does the Talaporfin Sodium patent expire?

No public expiry year is available for Talaporfin Sodium yet; this page updates once verified.

How many synthesis routes are recorded for Talaporfin Sodium?

2 synthesis routes are recorded; the shortest is 2 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Talaporfin Sodium intermediates?

All intermediates in Talaporfin Sodium routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Talaporfin Sodium intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-09-29