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Drugs Losing Exclusivity in 2029 & Key Intermediates

20 · Expiring drugs20 · Routes recorded20 · With on-sale intermediates

20 drugs expire in 2029 (public sources), 20 with recorded synthesis routes; key intermediates of 20 drugs are already available through the Unibest supply network. Generic developers typically secure intermediate supply 2–3 years ahead — use this table for shortlisting and RFQ.

DrugTierExpiryIndicationsRoutesCAS countAvailable
TicagrelorB · Position early2029Stroke, Acute coronary syndrome, Myocardial infarction555Available ×55
CarfilzomibB · Position early2029Multiple myeloma329Available ×29
Isavuconazonium SulfateC · Watch2029Mucorales infection, Aspergillus infection, Cryptosporidiosis122Available ×22
Cabozantinib S-malateB · Position early2029Neuroendocrine tumour, Pancreatic neuroendocrine tumour, Renal cell carcinoma321Available ×21
LinagliptinC · Watch2029Type 2 diabetes421Available ×21
Vonoprazan AcetateC · Watch2029Peptic ulcer bleeding420Available ×20
AbemaciclibA · Act now2029Breast cancer215Available ×15
Ribociclib SuccinateA · Act now2029Breast cancer114Available ×14
Dabrafenib MesylateB · Position early2029Thyroid cancer, Colorectal cancer, Glioma212Available ×12
TrametinibC · Watch2029Thyroid cancer, Glioma, Hairy cell leukaemia113Available ×6
Canagliflozin/Metformin HydrochlorideB · Position early2029End-stage renal disease, Cardiac and vascular disorders, Abdominal aortic aneurysm319Available ×5
BrexpiprazoleA · Act now2029Schizophrenia, Alzheimer's disease, Agitation312Available ×4
Cariprazine HydrochlorideA · Act now2029Major depressive disorder, Schizophrenia, Mania321Available ×4
Esketamine HydrochlorideB · Position early2029Major depressive disorder, Suicidal ideation, Depressive disorder836Available ×3
Pimavanserin TartrateC · Watch2029Delusion, Hallucination214Available ×3
DelafloxacinC · Watch2029Community-acquired bacterial pneumonia, Community-acquired pneumonia, Bacterial skin disease28Available ×3
AlpelisibC · Watch2029Growth disorder, Genetic disease, PIK3CA-related overgrowth spectrum217Available ×2
MirabegronB · Position early2029Neurogenic bladder dysfunction, Overactive bladder736Available ×1
Tedizolid PhosphateC · Watch2029Skin and skin structure infection, Staphylococcal infection, Bacterial skin disease322Available ×1
Cobimetinib FumarateC · Watch2029Melanoma330Available ×1

Frequently asked questions

Which drugs lose exclusivity in 2029?

20 drugs expire in 2029 per public sources: Abemaciclib, Ribociclib Succinate, Cabozantinib S-malate, Ticagrelor, Canagliflozin/Metformin Hydrochloride, Linagliptin, etc.

When should we start sourcing intermediates for 2029 launches?

Generic developers typically secure development-scale supply 2–3 years before expiry. 20 of the 20 drugs in this table already have on-sale intermediates in the Unibest network; the rest can be RFQ'd per CAS.

Are route and CAS data verified?

All fields are structured data cross-verified from public sources; intermediates carry registry codes and CAS numbers, and every "Available" badge links to real listings.

Source: cross-verified structured fields · Expiry years are public-source estimates; consult individual agencies for authoritative dates · 2026-09-29