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Drugs Losing Exclusivity in 2030 & Key Intermediates

19 · Expiring drugs18 · Routes recorded15 · With on-sale intermediates

19 drugs expire in 2030 (public sources), 18 with recorded synthesis routes; key intermediates of 15 drugs are already available through the Unibest supply network. Generic developers typically secure intermediate supply 2–3 years ahead — use this table for shortlisting and RFQ.

DrugTierExpiryIndicationsRoutesCAS countAvailable
FinerenoneC · Watch2030Systolic heart failure, Diastolic heart failure, Heart failure3596Available ×96
VenetoclaxB · Position early2030Acute myeloid leukaemia, Chronic lymphocytic leukaemia331Available ×31
Alectinib HydrochlorideB · Position early2030Non-small cell lung cancer, Lung cancer330Available ×30
ApalutamideA · Act now2030Castration-resistant prostate cancer, Prostate cancer220Available ×20
AcalabrutinibA · Act now2030Mantle cell lymphoma, Chronic lymphocytic leukaemia, Lymphocytic leukaemia214Available ×14
EntrectinibC · Watch2030Solid tumour, Non-small cell lung cancer114Available ×14
Mirogabalin besilateC · Watch2030Diabetic neuropathy, Postherpetic neuralgia, Peripheral nervous system disorder214Available ×14
Avatrombopag MaleateC · Watch2030Thrombocytopenia, Immune thrombocytopenic purpura, Liver disease111Available ×11
TucatinibC · Watch2030Breast cancer, Colorectal cancer110Available ×10
Dapagliflozin Propanediol/Metformin HydrochlorideA · Act now2030Type 2 diabetes416Available ×6
Neratinib MaleateC · Watch2030Breast cancer430Available ×3
EncorafenibC · Watch2030Non-small cell lung cancer, Colorectal cancer, Thyroid cancer123Available ×2
VadadustatC · Watch2030Chronic renal impairment, Anaemia212Available ×1
Omadacycline tosylateC · Watch2030Skin and skin structure infection, Community-acquired bacterial pneumonia, Bacterial infection314Available ×1
ErdafitinibC · Watch2030Urothelial carcinoma, Urinary tract neoplasm318Available ×1
LorlatinibB · Position early2030Non-small cell lung cancer220-
SelinexorC · Watch2030Diffuse large B-cell lymphoma, Multiple myeloma17-
Remimazolam BesilateC · Watch2030Sedation, Anaesthesia19-
EravacyclineC · Watch2030COVID-19---

Frequently asked questions

Which drugs lose exclusivity in 2030?

19 drugs expire in 2030 per public sources: Dapagliflozin Propanediol/Metformin Hydrochloride, Alectinib Hydrochloride, Lorlatinib, Venetoclax, Acalabrutinib, Entrectinib, etc.

When should we start sourcing intermediates for 2030 launches?

Generic developers typically secure development-scale supply 2–3 years before expiry. 15 of the 19 drugs in this table already have on-sale intermediates in the Unibest network; the rest can be RFQ'd per CAS.

Are route and CAS data verified?

All fields are structured data cross-verified from public sources; intermediates carry registry codes and CAS numbers, and every "Available" badge links to real listings.

Source: cross-verified structured fields · Expiry years are public-source estimates; consult individual agencies for authoritative dates · 2026-09-29