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CAS 1000889-99-5
(E)-4-chloro-2-(2-iodostyryl)phenol
Codes: ASEN-012-b
Application context (from source-drug indications)
SchizophreniaAsenapine MaleateManiaAsenapine MaleateBipolar I disorderAsenapine MaleateStutteringAsenapine MaleateParanoid schizophreniaAsenapine MaleateDisorganised schizophreniaAsenapine Maleate
Source drugs (routes using this intermediate)
| Drug | Tier | Expiry |
|---|---|---|
| Asenapine Maleate | Tier C — Watch / trade | - |
Position in synthesis routes (up/downstream chain)
Ordered by route registration; left → right is the synthesis direction. The highlighted node is the current CAS; others link to their own profiles.
5-chloro-2-hydroxybenzaldehyde→dimethylglycine→1-bromo-2-(bromomethyl)benzene→1-(chloromethyl)-2-iodobenzene→1-(bromomethyl)-2-chlorobenzene→diethyl (2-bromobenzyl)phosphonate→diethyl (2-iodobenzyl)phosphonate→diethyl (2-chlorobenzyl)phosphonate→(E)-2-(2-bromostyryl)-4-chlorophenol→(E)-4-chloro-2-(2-iodostyryl)phenol→(E)-4-chloro-2-(2-chlorostyryl)phenol→2-((3S,4S)-4-(2-bromophenyl)-1-methylpyrrolidin-3-yl)-4-chlorophenol→4-chloro-2-((3S,4S)-4-(2-iodophenyl)-1-methylpyrrolidin-3-yl)phenol→4-chloro-2-((3S,4S)-4-(2-chlorophenyl)-1-methylpyrrolidin-3-yl)phenol
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