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CAS 1644441-68-8

(Z)-methyl 4-(3-methoxy-1-((4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenyl)amino)-3-oxo-1-phenylprop-1-en-2-yl)-3-nitrobenzoate

Codes: NINT-025

Application context (from source-drug indications)

Systemic sclerosis-associated interstitial lung diseaseNintedanib EsylateIdiopathic pulmonary fibrosisNintedanib EsylateNon-small cell lung cancerNintedanib EsylatePulmonary fibrosisNintedanib EsylateInterstitial lung diseaseNintedanib EsylateHereditary haemorrhagic telangiectasiaNintedanib Esylate

Source drugs (routes using this intermediate)

DrugTierExpiry
Nintedanib EsylateTier B — Position early-

Position in synthesis routes (up/downstream chain)

Ordered by route registration; left → right is the synthesis direction. The highlighted node is the current CAS; others link to their own profiles.

Nintedanib EsylateOptimised routesteps: 3total yield: 2.37 g
methyl 4-(2-methoxy-2-oxoethyl)-3-nitrobenzoate→(trimethoxymethyl)benzene→N-(4-aminophenyl)-2-(4-methylpiperazin-1-yl)acetamide→(Z)-methyl 4-(1,3-dimethoxy-3-oxo-1-phenylprop-1-en-2-yl)-3-nitrobenzoate→(Z)-methyl 4-(3-methoxy-1-((4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenyl)amino)-3-oxo-1-phenylprop-1-en-2-yl)-3-nitrobenzoate

Intermediates available on this site

Side-by-side comparison of all listed offers on this CAS; price bands are list-price ranges, final price subject to RFQ confirmation.

SupplierProductPrice bandMOQLead timeQualificationsAction
Unibest Taizhou GMP-like Site2-Chloro-N-methyl-N-(4-nitrophenyl)acetamide
Pharmaceutical Intermediates
On requestOn requestOn request
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Qualified Partner — East China API WorksTrimethyl orthobenzoate
Pharmaceutical Intermediates
On requestOn requestOn request
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Unibest Nantong cGMP SiteN-(4-Aminophenyl)-N-methyl-2-(4-methylpiperazin -1-yl)acetamide
Pharmaceutical Intermediates
On requestOn requestOn request
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Unibest Taizhou GMP-like SiteMethyl 2-oxoindole-6-carboxylate
Pharmaceutical Intermediates
On requestOn requestOn request
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Qualified Partner — East China API Works(3E)-2,3-Dihydro-3-(methoxyphenylmethylene) -2-oxo-1H-indole-6- carboxylic acid methyl ester
Pharmaceutical Intermediates
On requestOn requestOn request
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This is a CAS-level registry record: registrations across routes are merged. Supplier offers and buyer demands will be matched on this CAS as the primary key.