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CAS 106910-77-4

N-Benzyl-D-serine

Codes: (I)448314-2-a

Application context (from source-drug indications)

Hot flushesElinzanetantVasomotor symptomsElinzanetantHR阳性乳腺癌Elinzanetant睡眠障碍ElinzanetantMenopausal symptomsElinzanetantOpioid dependenceElinzanetant

Source drugs (routes using this intermediate)

DrugTierExpiry
ElinzanetantTier C — Watch / trade-

Position in synthesis routes (up/downstream chain)

Ordered by route registration; left → right is the synthesis direction. The highlighted node is the current CAS; others link to their own profiles.

ElinzanetantOptimised routesteps: 10total yield: /
N-Benzyl-D-serine→2-Chloranylethanoyl chloride→4-Benzyl-5-oxomorpholine-3(R)-carboxylic acid→[(3S)-4-Benzylmorpholin-3-yl]methanol hydrogen chloride (1/1)→[(3S)-Morpholin-3-yl]methanol hydrogen chloride (1/1)→3-(Benzyloxy)-2(R)-(tert-butoxycarbonylamino)propionic acid→tert-Butyl [(2R)-3-(benzyloxy)-1-[(3S)-3-(hydroxymethyl)morpholin-4-yl]-1-oxopropan-2-yl]carbamate→tert-Butyl [(2S)-1-(benzyloxy)-3-[(3S)-3-(hydroxymethyl)morpholin-4-yl]propan-2-yl]carbamate→tert-Butyl [(2S)-1-(benzyloxy)-3-[(3R)-3-(chloromethyl)morpholin-4-yl]propan-2-yl]carbamate→(2S)-1-(Benzyloxy)-3-[(3R)-3-(chloromethyl)morpholin-4-yl]propan-2-amine→(7S,9aS)-7-[(Benzyloxy)methyl]octahydropyrazino[2,1-c][1,4]oxazine→2-[3,5-Bis(trifluoromethyl)phenyl]-N-[6-chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-yl]-N,2-dimethylpropanamide→N-[6-[(7S,9aS)-7-[(Benzyloxy)methyl]hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-4-(4-fluoro-2-methylphenyl)pyridin-3-yl]-2-[3,5-bis(trifluoromethyl)phenyl]-N,2-dimethylpropanamide hydrogen chloride (1/2)→N-[6-[(7S,9aS)-7-[(Benzyloxy)methyl]hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]-4-(4-fluoro-2-methylphenyl)pyridin-3-yl]-2-[3,5-bis(trifluoromethyl)phenyl]-N,2-dimethylpropanamide

Intermediates available on this site

Side-by-side comparison of all listed offers on this CAS; price bands are list-price ranges, final price subject to RFQ confirmation.

SupplierProductPrice bandMOQLead timeQualificationsAction
Unibest Taizhou GMP-like SiteN-Boc-O-Benzyl-D-serine
Pharmaceutical Intermediates
On requestOn requestOn request
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Qualified Partner — East China API Works6-chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-amine hydrochloride
Pharmaceutical Intermediates
On requestOn requestOn request
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Unibest Nantong cGMP SiteN-[6-Chloro-4-(4-fluoro-2-methylp henyl)-3-pyridinyl]-N,a,a-trimethy
Pharmaceutical Intermediates
On requestOn requestOn request
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Unibest Taizhou GMP-like Site3-Morpholinemethanol, 4-(phenylmethyl)-, hydrochloride
Pharmaceutical Intermediates
On requestOn requestOn request
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Qualified Partner — East China API Works(7S,9aS)-7-((Benzyloxy)methyl)octahydropyrazino[2,1-c][1,4]oxazine dioxalate salt
Pharmaceutical Intermediates
On requestOn requestOn request
—
Unibest Nantong cGMP Site2-(3,5-bis(trifluoroMethyl)phenyl)-2-Methyl propanoic acid
Pharmaceutical Intermediates
On requestOn requestOn request
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Unibest Taizhou GMP-like Site((7S)-octahydropyrazino[2,1-c][1,4]oxazin-7-yl)methanol
Pharmaceutical Intermediates
On requestOn requestOn request
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Qualified Partner — East China API Works4-Boc-3-morpholinecarboxylic Acid
Pharmaceutical Intermediates
On requestOn requestOn request
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Unibest Nantong cGMP Site2-(3,5-bis-trifluoromethylphenyl)-2-methyl-propionyl chloride
Pharmaceutical Intermediates
On requestOn requestOn request
—

This is a CAS-level registry record: registrations across routes are merged. Supplier offers and buyer demands will be matched on this CAS as the primary key.